XAV-939 CAS:284028-89-3
XAV-939
Catalog # | Pkg Size | Price(USD) | Quantity | Buy this product |
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R-C-2663 | 100mg | 300.00 | + Add to cart |
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R-C-2663 | 200mg | 520.00 | + Add to cart |
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R-C-2663 | 500mg | 720.00 | + Add to cart |
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Product description
XAV-939 is a potent tankyrase inhibitor that targets Wnt/β-catenin signaling.XAV-939 stabilizes axin by inhibiting tankyrase 1 and tankyrase 2(IC50s of 5 and 2nM,respectively),thereby stimulating β-catenin degradation.XAV939 binds tightly to the catalytic(PARP)domains of TNKS1 and TNKS2(Kds of 99 and 93nM,respectively).
Appearance | N/A |
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Molecular Weight | N/A |
purity | >95% |
PDI by GPC | N/A |
Solubility | N/A |
Storage | -20℃, protected from light and moisture |
Transportation | 4-25℃ temperature for up to 3 weeks |
Stability | 2 years |
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